Tacrine (Cognex) -|- Pharmacology Mnemonics - Flash Cards

Tacrine (Cognex)

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Name: Tacrine (Cognex)

Class: Anticholinesterase Agent: Acridinamine

Mech.: Blocks AChE and BuChE. Inhib. M1 and M2 receptors. Weak nicotinic blocker. ­ release of ACh from nerve endings.

Absorption:

Dist.: Good CNS.

Metab.:

Excretion, :

Toxicity/S.E.s: Reversible liver damage. Avoid in cases of asthma, coronary insufficiency, peptic ulcers.

Utility: Alzheimer’s disease

Special Features: